BDBM50049806 CHEMBL127969::Thiophene-2-carboxylic acid [2-(1-methyl-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-2-yl)-ethyl]-amide
SMILES CN1C(CCNC(=O)c2cccs2)CN=C(c2ccccc2)c2ccccc12
InChI Key InChIKey=PYCHFYLMMMZMSJ-UHFFFAOYSA-N
Data 10 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50049806
Affinity DataKi: 0.5nMAssay Description:Binding affinity against Opioid receptor kappa 1 of guinea pig using [3H]-U-65,693 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding affinity against Opioid receptor mu 1 using [3H]-DAMGO as radioligand in guinea pig brainMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding affinity of compound was determined against Opioid receptor mu 1 from native receptor in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Binding affinity determined against Opioid receptor mu 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Binding affinity determined against Opioid receptor delta 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Binding affinity against Opioid receptor delta 1 using [3H]-DADLE as radioligand in guinea pig brainMore data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Binding affinity of compound was determined against Opioid receptor delta 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Binding affinity against Cholecystokinin type B receptor using [3H](MeNLE28,31)-CCK-8 as radioligand in guinea pig cerebral cortex.More data for this Ligand-Target Pair