BDBM50057509 (2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1-methyl-1,4,5,6-tetrahydro-2H-benzo[e][1,4]diazocin-3-one::8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1-methyl-1,4,5,6-tetrahydro-2H-benzo[e][1,4]diazocin-3-one::CHEMBL6453
SMILES CCCCCCCCC#Cc1ccc2N(C)[C@@H](C(C)C)C(=O)N[C@H](CO)Cc2c1
InChI Key InChIKey=KDIRIFZBLUSLJU-UPVQGACJSA-N
Data 19 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 19 hits for monomerid = 50057509
Affinity DataKi: 6.15nMAssay Description:Binding affinity against RAS guanyl releasing protein using [3H]- PDBu as the labeled ligandMore data for this Ligand-Target Pair
Affinity DataKi: 10.7nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of [3H]-PDBu binding to PKC delta wild typeMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC alpha expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of phorbol 12,13-dibutyrate (PDBU) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 17.4nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC beta expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C alphaMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C epsilonMore data for this Ligand-Target Pair
Affinity DataKi: 40.7nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C betaMore data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 122nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC delta expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 134nMAssay Description:Inhibition of [3H]-PDBu binding to PKC delta mutant Leu 20-GlyMore data for this Ligand-Target Pair
Affinity DataKi: 142nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC epsilon expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 730nMAssay Description:Inhibition of [3H]-PDBu binding to PKC delta mutant Pro 11-GlyMore data for this Ligand-Target Pair
Affinity DataKi: 933nMAssay Description:Inhibition of [3H]-PDBu binding to PKC delta mutant Gln 27-ValMore data for this Ligand-Target Pair