BDBM50074353 (2-Bromo-4,6-dimethoxy-phenyl)-ethyl-(4-methyl-6-morpholin-4-yl-[1,3,5]triazin-2-yl)-amine::CHEMBL424204::CHEMBL43216

SMILES CCN(c1nc(C)nc(n1)N1CCOCC1)c1c(Br)cc(OC)cc1OC

InChI Key InChIKey=FKWFEXHQWCTXFD-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50074353   

TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50074353((2-Bromo-4,6-dimethoxy-phenyl)-ethyl-(4-methyl-6-m...)
Affinity DataKi:  32nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50074353((2-Bromo-4,6-dimethoxy-phenyl)-ethyl-(4-methyl-6-m...)
Affinity DataKi:  32nMAssay Description:Inhibition of binding of the radioligand, [125 I-Tyr0]-CRF to rat cerebral cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50074353((2-Bromo-4,6-dimethoxy-phenyl)-ethyl-(4-methyl-6-m...)
Affinity DataKi:  43nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed