BDBM50088002 1-(4-carboxymethoxyphenyl)-11-[2-(2-methoxyphenyl)acryloyl]-(1R,8R,9S,13S)-11-azatetracyclo[6.5.2.02,7.09,13]pentadeca-2,4,6-triene-9-carboxylic acid (RPR132506)::CHEMBL297030

SMILES C=C(C(=O)N1C[C@H]2[C@@]3(c4ccc(OCC(=O)O)cc4)CC[C@H](c4ccccc43)[C@@]2(C(=O)O)C1)c1ccccc1OC

InChI Key InChIKey=LENBZZVPKVZQEV-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50088002   

TargetDimer of Protein farnesyltransferase subunit beta(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50088002BDBM50088002(1-(4-carboxymethoxyphenyl)-11-[2-(2-methoxyphenyl)...)
Affinity DataKi:  2.55E+4nMAssay Description:Inhibition of farnesyltransferase by Ras/SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed