BDBM50097789 2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imidazo[1,2-a]pyrazin-2-yl]-N-cyclohexyl-isobutyramide::CHEMBL165402

SMILES CC(C)(C(=O)NC1CCCCC1)c1cn2cc(nc(CCCN)c2n1)-c1csc2ccccc12

InChI Key InChIKey=QSIQDAIODXAVEF-UHFFFAOYSA-N

Data  5 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50097789   

TargetSomatostatin receptor type 5(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50097789(2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imid...)
Affinity DataKi:  360nMAssay Description:Inhibitory constant on human somatostatin receptor 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50097789(2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imid...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity on human somatostatin receptor 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50097789(2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imid...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibitory constant on human somatostatin receptor type 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50097789(2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imid...)
Affinity DataKi:  9.50E+3nMAssay Description:Inhibitory constant on human Somatostatin receptor type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50097789(2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imid...)
Affinity DataKi:  9.70E+3nMAssay Description:Inhibitory constant on human Somatostatin receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50097789(2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imid...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant on human somatostatin receptor 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed