BDBM50099173 2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine::CHEMBL175197

SMILES NC(=N[C@H](Cc1c[nH]c2ccccc12)c1nc(c[nH]1)-c1ccccc1)c1ccc(F)cc1F

InChI Key InChIKey=MTBMFGLKEXFYMH-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50099173   

TargetSomatostatin receptor type 3(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50099173(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
Affinity DataKi:  200nMAssay Description:Inhibition of human sst3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50099173(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibition of human sst1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50099173(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
Affinity DataKi:  2.25E+3nMAssay Description:Inhibition of human sst5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50099173(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human sst2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50099173(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human sst4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed