BDBM50100746 CHEMBL265912::Des-AA1,2,4,5,12,13-[DTrp8]-SRIF

SMILES C[C@@H](O)[C@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](N)CSSC[C@H](NC(=O)[C@H](Cc2ccccc2)NC1=O)C(O)=O

InChI Key InChIKey=PJRZZHKHLDKTKL-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50100746   

TargetSomatostatin receptor type 4(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100746(Des-AA1,2,4,5,12,13-[DTrp8]-SRIF | CHEMBL265912)
Affinity DataIC50: 1.30nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100746(Des-AA1,2,4,5,12,13-[DTrp8]-SRIF | CHEMBL265912)
Affinity DataIC50: 13.1nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100746(Des-AA1,2,4,5,12,13-[DTrp8]-SRIF | CHEMBL265912)
Affinity DataIC50: 27.3nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100746(Des-AA1,2,4,5,12,13-[DTrp8]-SRIF | CHEMBL265912)
Affinity DataIC50: 43.8nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100746(Des-AA1,2,4,5,12,13-[DTrp8]-SRIF | CHEMBL265912)
Affinity DataIC50: 45.7nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed