BDBM50122253 CHEMBL3617639

SMILES COc1cccc(c1)N1C[C@@H](C)n2nc(COc3ccc(Cl)cn3)cc2C1=O

InChI Key InChIKey=HDKXWARCXQYIAT-CYBMUJFWSA-N

Data  2 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50122253   

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122253(CHEMBL3617639)
Affinity DataIC50:  316nMAssay Description:Negative allosteric modulation of rat mGlu3 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122253(CHEMBL3617639)
Affinity DataEC50:  5.13E+3nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122253(CHEMBL3617639)
Affinity DataEC50:  5.07E+3nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122253(CHEMBL3617639)
Affinity DataIC50:  313nMAssay Description:Negative allosteric modulation of rat mGlu3 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed