BDBM50124609 5-Allyl-2,2,4-trimethyl-10-prop-2-ynyloxy-2,5-dihydro-1H-6-oxa-1-aza-chrysene::CHEMBL8360
SMILES CC1=CC(C)(C)Nc2ccc-3c(C(CC=C)Oc4cccc(OCC#C)c-34)c12
InChI Key InChIKey=SNHVWFHHKLONNR-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50124609
Affinity DataKi: 4.20nMAssay Description:Binding affinity towards human glucocorticoid receptor (GR) was determined using [3H]-Dexamethasone as radioligand in SF-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >300nMAssay Description:Transcriptional repression in HepG2 cells expressing human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Binding affinity towards aldosterone receptor (Mineralocorticoid receptor)More data for this Ligand-Target Pair