BDBM50128276 CHEMBL3628725

SMILES Cn1cc(c(n1)-c1ccc(OCc2ccc3cc(CF)ccc3n2)cc1)-c1ccncc1

InChI Key InChIKey=GOOCZSKXXSGRFQ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50128276   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Washington University

Curated by ChEMBL

LigandBDBM50128276(CHEMBL3628725)Copy SMILESCopy InChI

Affinity DataIC50: 76nMAssay Description:Inhibition of recombinant human PDE10A assessed as reduction of [3H]-cAMP hydrolysis preincubated for 5 mins followed by [3H]-cAMP addition measured ...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
12/15/2016
Entry Details Article
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