BDBM50129663 3-But-3-enoylamino-pyridine-2-carboxylic acid thiazol-2-ylamide::CHEMBL90048

SMILES C=CCC(=O)Nc1cccnc1C(=O)Nc1nccs1

InChI Key InChIKey=WAPRPWZOYLYCTM-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50129663   

TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50129663(3-But-3-enoylamino-pyridine-2-carboxylic acid thia...)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibitory concentration required against Escherichia coli MetAP1 (150 nM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Baker's yeast)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50129663(3-But-3-enoylamino-pyridine-2-carboxylic acid thia...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50129663(3-But-3-enoylamino-pyridine-2-carboxylic acid thia...)
Affinity DataIC50:  130nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed