BDBM50130275 4-(3-(2-(dimethylamino)ethyl)-1H-indol-1-ylsulfonyl)benzenamine::4-[3-(2-Dimethylamino-ethyl)-indole-1-sulfonyl]-phenylamine::4-{3-[2-(dimethylamino)ethyl]-1H-indole-1-sulfonyl}aniline, 7::CHEMBL94093

SMILES CN(C)CCc1cn(c2ccccc12)S(=O)(=O)c1ccc(N)cc1

InChI Key InChIKey=FBZNHEBASSSMLO-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50130275   

Target5-hydroxytryptamine receptor 6(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50130275(4-{3-[2-(dimethylamino)ethyl]-1H-indole-1-sulfonyl...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50130275(4-{3-[2-(dimethylamino)ethyl]-1H-indole-1-sulfonyl...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H] LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50130275(4-{3-[2-(dimethylamino)ethyl]-1H-indole-1-sulfonyl...)
Affinity DataKi:  0.800nMpH: 7.4Assay Description:The h5-HT6 radioligand binding assays were performed as previously described. In brief, h5-HT6 cDNA was transiently expressed in HEK-293 cells using...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2013
Entry Details Article

Target5-hydroxytryptamine receptor 6(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50130275(4-{3-[2-(dimethylamino)ethyl]-1H-indole-1-sulfonyl...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed