BDBM50133229 1-Methyl-2-(3,7,8,9-tetrahydro-pyrano[3,2-e]indol-1-yl)-ethylamine::CHEMBL133868
SMILES CC(N)Cc1c[nH]c2ccc3OCCCc3c12
InChI Key InChIKey=VVHJUSGIUWQPIT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 22 hits for monomerid = 50133229
Affinity DataKi: 0.300nMAssay Description:In vitro inhibitory constant against [125I]DOI binding to 5-hydroxytryptamine 2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibitory constant against cloned human 5-hydroxytryptamine 2A receptor using with [125I]- DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibitory constant against cloned human 5-hydroxytryptamine 2C receptor using with [125I]- DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory constant against cloned human 5-hydroxytryptamine 2B receptor using with [125I]- DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Inhibitory constant against human 5-hydroxytryptamine 6 receptor using [3H]LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Inhibitory constant against 5-hydroxytryptamine 4 receptor using [3H]GR-113808 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Inhibitory constant against human 5-hydroxytryptamine 5A receptor using [3H]LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Inhibitory constant against Alpha-2B adrenergic receptor using [3H]MK-912 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against human 5-hydroxytryptamine 1B receptor using [3H]5-CT radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against human serotonin transporter using [3H]N-Me-citalopram radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against 5-hydroxytryptamine 3 receptor using [3H]GR-65630 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against 5-hydroxytryptamine 1B receptor using with [125I]- cyanopindolol radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Inhibitory constant against human 5-hydroxytryptamine 7 receptor using [3H]LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory constant against Alpha-1A adrenergic receptor using [3H]-7-MeO prazosin radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory constant against norepinephrine transporter receptor using [3H]radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory constant against Alpha-1B adrenergic receptor using [3H]-7-MeO prazosin radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+4nMAssay Description:In vitro inhibitory concentration required against [3H]8-OH-DPAT binding to cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 116nMAssay Description:In vitro relative agonist activity against 5-hydroxytryptamine 2A using PI assay in rat vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for functional response on CHO cells expressing cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration required against Alpha-2A adrenergic receptor using [3H]clonidine radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibition of [125I]DOI binding to 5-hydroxytryptamine 2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory concentration required against Alpha-2C adrenergic receptor using [3H]clonidine radioligandMore data for this Ligand-Target Pair