BDBM50133363 CHEMBL541455::N-(2-(furan-2-yl)-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-phenylacetamide::N-(2-Furan-2-yl-8-phenethyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-2-phenyl-acetamide
SMILES O=C(Cc1ccccc1)Nc1nc2nn(CCc3ccccc3)cc2c2nc(nn12)-c1ccco1
InChI Key InChIKey=NNKNPNUOGFMYAG-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50133363
Affinity DataKi: 5.49nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 43.9nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Displacement of [3H]-MRE3008-F20 from human A3 receptors expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]-ZM-241,385 from human adenosine A2A receptors expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 128nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced adenylyl cyclase activityChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair