BDBM50134310 9-Methoxy-2-methyl-2,3,10,10a-tetrahydro-pyrazino[1,2-a]indole-1,4-dione::CHEMBL333703

SMILES COc1cccc2N3C(Cc12)C(=O)N(C)CC3=O

InChI Key InChIKey=ZJOTVAYTCJHWQQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50134310   

LigandPNGBDBM50134310(9-Methoxy-2-methyl-2,3,10,10a-tetrahydro-pyrazino[...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134310(9-Methoxy-2-methyl-2,3,10,10a-tetrahydro-pyrazino[...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras-CVLS by farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed