BDBM50136420 5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyridin-3-ylmethyl-1,2,3,4-tetrahydro-quinolin-3-yl)-amide::CHEMBL136567

SMILES O=C(NC1Cc2ccccc2N(Cc2cccnc2)C1=O)c1cc2cc(Cl)ccc2[nH]1

InChI Key InChIKey=PUCJVQSSYZACPP-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50136420   

TargetGlycogen phosphorylase, liver form(Human)
Applied Science University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50136420BDBM50136420(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyri...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Applied Science University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50136420BDBM50136420(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyri...)
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed