BDBM50139019 (S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(1S,2R)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-phenyl-propyl]-amide::CHEMBL423794
SMILES C[C@@H]([C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(N)=O)c1ccccc1
InChI Key InChIKey=GHCQVWCTWHWODK-GYZIEVATSA-N
Data 5 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50139019
TargetMu-type opioid receptor(Rat)
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [3H]-endomorphin-2 from Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rat)
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 55.7nMAssay Description:Displacement of [3H]-Dynorphin A from Opioid receptor kappa 1 of rat brain membranes (DAMGO/DADLE quenching of mu/delta receptor binding)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 106nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 106nMAssay Description:Displacement of [3H]-DAMGO from Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rat)
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ile5,6-deltorphin II from opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair