BDBM50139574 4-{5-[(3-Oxo-2-phenyl-2,3,4,5-tetrahydro-1H-benzo[c]azepin-4-ylamino)-methyl]-imidazol-1-ylmethyl}-benzonitrile::CHEMBL162968

SMILES O=C1C(Cc2ccccc2CN1c1ccccc1)NCc1cncn1Cc1ccc(cc1)C#N

InChI Key InChIKey=DZJIZUHWPKFMQZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50139574   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50139574(4-{5-[(3-Oxo-2-phenyl-2,3,4,5-tetrahydro-1H-benzo[...)
Affinity DataIC50:  26nMAssay Description:Inhibition of farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed