BDBM50139586 4-(5-{[3-(3,5-Difluoro-benzyl)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[d]azepin-1-ylamino]-methyl}-imidazol-1-ylmethyl)-benzonitrile::CHEMBL165519

SMILES Fc1cc(F)cc(CN2CCc3ccccc3C(NCc3cncn3Cc3ccc(cc3)C#N)C2=O)c1

InChI Key InChIKey=VXXYAJGHLFTFPE-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50139586   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Human)
Institut De Recherches Servier

Curated by ChEMBL

LigandBDBM50139586(4-(5-{[3-(3,5-Difluoro-benzyl)-2-oxo-2,3,4,5-tetra...)Copy SMILESCopy InChI

Affinity DataIC50: 26nMAssay Description:Inhibition of farnesyltransferaseMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/10/2009
Entry Details Article
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