BDBM50139590 4-(5-{[3-Oxo-2-(2,3,5-trifluoro-benzyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-4-ylamino]-methyl}-imidazol-1-ylmethyl)-benzonitrile::CHEMBL164286

SMILES Fc1cc(F)c(F)c(CN2Cc3ccccc3CC(NCc3cncn3Cc3ccc(cc3)C#N)C2=O)c1

InChI Key InChIKey=SSYAXKLPIZZQEY-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50139590   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Human)
Institut De Recherches Servier

Curated by ChEMBL

LigandBDBM50139590(4-(5-{[3-Oxo-2-(2,3,5-trifluoro-benzyl)-2,3,4,5-te...)Copy SMILESCopy InChI

Affinity DataIC50: 18nMAssay Description:Inhibition of farnesyltransferaseMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/10/2009
Entry Details Article
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