BDBM50150326 4-[4-(4-{[Benzyl-(3-methanesulfonylamino-2-methyl-phenyl)-amino]-methyl}-phenoxy)-phenyl]-butyric acid::CHEMBL182496

SMILES Cc1c(NS(C)(=O)=O)cccc1N(Cc1ccccc1)Cc1ccc(Oc2ccc(CCCC(O)=O)cc2)cc1

InChI Key InChIKey=DVRXYXZNRPMKQA-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50150326   

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50150326(4-[4-(4-{[Benzyl-(3-methanesulfonylamino-2-methyl-...)
Affinity DataIC50:  670nMAssay Description:Inhibition of glucocorticoid receptor dexamethasone responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50150326(4-[4-(4-{[Benzyl-(3-methanesulfonylamino-2-methyl-...)
Affinity DataIC50:  670nMAssay Description:Inhibition of glucocorticoid receptor Dexamethasone response in reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50150326(4-[4-(4-{[Benzyl-(3-methanesulfonylamino-2-methyl-...)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of [3H]dexamethasone binding to human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50150326(4-[4-(4-{[Benzyl-(3-methanesulfonylamino-2-methyl-...)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of [3H]-dexamethasone binding to glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed