BDBM50151849 CHEMBL3774907

SMILES c1ccc(Nc2nc(-c3cccc4[nH]ncc34)nc(N3CCOCC3)n2)cc1

InChI Key InChIKey=ASOLRIGVQKJPHG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50151849   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Sphaera Pharma

Curated by ChEMBL

LigandBDBM50151849(CHEMBL3774907)Copy SMILESCopy InChI

Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant PI3K-alpha using phosphatidylinositol biphosphate as substrate preincubated for 15 mins followed by substrate additio...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
7/1/2017
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL