BDBM50152467 8-{1-Methyl-2-[(thiophen-3-ylmethyl)-amino]-ethoxy}-quinolin-2-ylamine::CHEMBL187847

SMILES CC(CNCc1ccsc1)Oc1cccc2ccc(N)nc12

InChI Key InChIKey=KUOMQPQUGJCJDT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50152467   

TargetMelanin-concentrating hormone receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50152467(8-{1-Methyl-2-[(thiophen-3-ylmethyl)-amino]-ethoxy...)
Affinity DataIC50: 10nMAssay Description:Concentration required to inhibit binding of [125I]-MCH radioligand to human Melanin-concentrating hormone receptor 1 in IMR-32 I3.4.2 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed