BDBM50153453 3-[1-(4-Dimethylamino-butyl)-1H-indol-3-yl]-4-phenylamino-pyrrole-2,5-dione::CHEMBL184548

SMILES CN(C)CCCCn1cc(C2=C(Nc3ccccc3)C(=O)NC2=O)c2ccccc12

InChI Key InChIKey=XULMLPZWWAPYHV-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50153453   

TargetProtein kinase C alpha type(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153453(3-[1-(4-Dimethylamino-butyl)-1H-indol-3-yl]-4-phen...)
Affinity DataIC50:  730nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C epsilon type(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153453(3-[1-(4-Dimethylamino-butyl)-1H-indol-3-yl]-4-phen...)
Affinity DataIC50:  5.87E+3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C epsilonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50153453(3-[1-(4-Dimethylamino-butyl)-1H-indol-3-yl]-4-phen...)
Affinity DataIC50:  15nMAssay Description:Inhibition of PKCbeta2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50153453(3-[1-(4-Dimethylamino-butyl)-1H-indol-3-yl]-4-phen...)
Affinity DataIC50:  15nMAssay Description:Inhibition of PKCbeta2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50153453(3-[1-(4-Dimethylamino-butyl)-1H-indol-3-yl]-4-phen...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C beta 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed