BDBM50156861 2-(2-(4-(1-((5-chlorothiophen-2-yl)methyl)-6-fluoro-1H-indol-3-yl)piperidin-1-yl)ethoxy)benzoic acid::CHEMBL374459

SMILES OC(=O)c1ccccc1OCCN1CCC(CC1)c1cn(Cc2ccc(Cl)s2)c2cc(F)ccc12

InChI Key InChIKey=XKAJSRFEDJSVQV-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50156861   

TargetHistamine H2 receptor(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156861(2-(2-(4-(1-((5-chlorothiophen-2-yl)methyl)-6-fluor...)
Affinity DataIC50:  1.03E+3nMAssay Description:Displacement of [3H]ketanserine from histamine H2 receptor in human cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156861(2-(2-(4-(1-((5-chlorothiophen-2-yl)methyl)-6-fluor...)
Affinity DataIC50:  28nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed