BDBM50156862 4-bromo-3-((4-(1-(2-ethoxyethyl)-1H-indol-3-yl)piperidin-1-yl)methyl)benzoic acid::CHEMBL222214

SMILES CCOCCn1cc(C2CCN(Cc3cc(ccc3Br)C(O)=O)CC2)c2ccccc12

InChI Key InChIKey=RPSZKBDNKHVSEN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50156862   

TargetHistamine H2 receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156862(4-bromo-3-((4-(1-(2-ethoxyethyl)-1H-indol-3-yl)pip...)
Affinity DataIC50:  5.60E+3nMAssay Description:Displacement of [3H]ketanserine from histamine H2 receptor in human cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156862(4-bromo-3-((4-(1-(2-ethoxyethyl)-1H-indol-3-yl)pip...)
Affinity DataIC50:  345nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed