BDBM50156879 2-{2-[4-(1-butyl-6-fluoro-1H-indol-3-yl)piperidin-1-yl]-ethoxy}benzoic acid::CHEMBL221664

SMILES CCCCn1cc(C2CCN(CCOc3ccccc3C(O)=O)CC2)c2ccc(F)cc12

InChI Key InChIKey=ZMOAWDWBPDLQAJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50156879   

TargetHistamine H2 receptor(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156879(2-{2-[4-(1-butyl-6-fluoro-1H-indol-3-yl)piperidin-...)
Affinity DataIC50:  2.15E+3nMAssay Description:Displacement of [3H]ketanserine from histamine H2 receptor in human cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156879(2-{2-[4-(1-butyl-6-fluoro-1H-indol-3-yl)piperidin-...)
Affinity DataIC50:  47nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed