BDBM50156884 3-[4-(1-thiophen-2-ylmethyl-1H-indol-3-yl)piperidin-1-ylmethyl]benzoic acid::CHEMBL222372

SMILES OC(=O)c1cccc(CN2CCC(CC2)c2cn(Cc3cccs3)c3ccccc23)c1

InChI Key InChIKey=IZCYYVKHBBLUDY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50156884   

TargetHistamine H1 receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156884(3-[4-(1-thiophen-2-ylmethyl-1H-indol-3-yl)piperidi...)
Affinity DataIC50:  90nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50156884(3-[4-(1-thiophen-2-ylmethyl-1H-indol-3-yl)piperidi...)
Affinity DataIC50:  1.33E+3nMAssay Description:Displacement of [3H]ketanserine from histamine H2 receptor in human cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed