BDBM50157607 CHEMBL3753082::US11773085, Compound B24
SMILES CC(C)CS(=O)(=O)N[C@H]1CCC(=O)N([C@@H]1c1ccc(Cl)cc1)c1ccc2c(C)cc(=O)n(C)c2c1
InChI Key InChIKey=LVDRREOUMKACNJ-BKMJKUGQSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 14 hits for monomerid = 50157607
Affinity DataKd: 99nMAssay Description:Binding affinity to BRD9 (unknown origin) by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human BRD9 isoform 1 co-expressed with H4 histone in HEK293 cells preincubated for 18 hrs followed by addition of nano-BRET furimazine ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human BRD9 isoform 1 co-expressed with H3 histone family 3A in HEK293 cells preincubated for 18 hrs followed by addition of nano-BRET f...More data for this Ligand-Target Pair
Affinity DataKd: 909nMAssay Description:Inhibition of human BRD7 by VP-ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 99nMAssay Description:Inhibition of human BRD9 isoform 1 by VP-ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 909nMAssay Description:Binding affinity to human BRD7 by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 909nMAssay Description:Inhibition of BRD7 (unknown origin) by Isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 99nMAssay Description:Binding affinity to recombinant human BRD9 by isothermal calorimetric titration methodMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity to BRD7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to BRD9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 99nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:A mixture of biotinylated-ligand and SureLight Allophycocyanin-Streptavidin (APC-SA, PerkinElmer AD0201) in 50 mM HEPES (pH 7.4), 50 mM NaCl, 1 mM TC...More data for this Ligand-Target Pair
Affinity DataKd: 99nMAssay Description:Inhibition of BRD9 (unknown origin) by Isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 99nMAssay Description:Binding affinity to human BRD9 by ITC analysisMore data for this Ligand-Target Pair