BDBM50162083 (5-Methyl-1H-pyrazol-3-yl)-(2-phenyl-quinazolin-4-yl)-amine::(5-Methyl-1H-pyrazol-3-yl)-(2-phenylquinazolin-4-yl)amine::CHEMBL359482::N-(3-methyl-1H-pyrazol-5-yl)-2-phenylquinazolin-4-amine::N-(5-METHYL-1H-PYRAZOL-3-YL)-2-PHENYLQUINAZOLIN-4-AMINE
SMILES Cc1cc(Nc2nc(nc3ccccc23)-c2ccccc2)[nH]n1
InChI Key InChIKey=JYCUVOXSZBECAY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50162083
Affinity DataKi: 22nMAssay Description:Inhibition of Gsk3betaChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of Glycogen synthase kinase-3More data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Inhibition of Aurora-A by coupled assayMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Inhibition of aurora A kinaseChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Inhibition of SrcChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 858nMAssay Description:Inhibition of Aurora B (unknown origin) using FAM-labelled peptide as substrate pretreated for 10 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of Aurora A (unknown origin) using FAM-labelled peptide as substrate pretreated for 10 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase(Human)
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human recombinant PKR autophosphorylation using poly[I:C] after 10 mins by luminescent assayMore data for this Ligand-Target Pair