BDBM50168665 CHEMBL185625::N-(1-{4-[(R)-2-(3-Amino-propionylamino)-3-(2,4-dichloro-phenyl)-propionyl]-piperazin-1-yl}-cyclohexylmethyl)-4-trifluoromethoxy-benzamide

SMILES NCCC(=O)N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)N1CCN(CC1)C1(CNC(=O)c2ccc(OC(F)(F)F)cc2)CCCCC1

InChI Key InChIKey=PHDZAKCPWCXBFC-AREMUKBSSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50168665   

TargetMelanocortin receptor 4(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50168665(CHEMBL185625 | N-(1-{4-[(R)-2-(3-Amino-propionylam...)
Affinity DataKi:  400nMAssay Description:Inhibition of [125I]-AgRP(83132) (radioligand) binding to the hMC4R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed