BDBM50172073 CHEMBL3809509

SMILES C[C@@H](OC(=O)N1CCC2(CC1)CCc1cc(ccc1O2)-c1ccc(CS(=O)(=O)Cc2ccccn2)cc1)C(F)(F)F

InChI Key InChIKey=BPSYRTWSVUOMPE-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50172073   

TargetGlucose-dependent insulinotropic receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50172073(CHEMBL3809509)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human GPR119 receptor assessed as increase in cellular cAMP levels by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2017
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50172073(CHEMBL3809509)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human GPR119 expressed in CHO-K1 cells after 4 hrs by Bright-Glo luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed