BDBM50173188 CHEMBL383568::[4-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin-6-yl)-phenyl]-morpholin-4-yl-methanone

SMILES Nc1nc(cn2nc(nc12)-c1ccco1)-c1ccc(cc1)C(=O)N1CCOCC1

InChI Key InChIKey=HBJDPRRWVDNJBD-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50173188   

TargetAdenosine receptor A2a(Rat)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50173188(CHEMBL383568 | [4-(8-Amino-2-furan-2-yl-[1,2,4]tri...)
Affinity DataKi:  19nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50173188(CHEMBL383568 | [4-(8-Amino-2-furan-2-yl-[1,2,4]tri...)
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity towards adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX compared to SCH-58261 (Ki=390 nM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed