BDBM50175109 CHEMBL199649::N-(2,4-dimethoxyphenethyl)oleamide

SMILES CCCCCCCC\C=C/CCCCCCCC(=O)NCCc1ccc(OC)cc1OC

InChI Key InChIKey=YDMFQRINHJCRDN-UHFFFAOYSA-N

Data  3 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50175109   

TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175109(N-(2,4-dimethoxyphenethyl)oleamide | CHEMBL199649)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor in presence of hydrolase inhibitor PMSFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175109(N-(2,4-dimethoxyphenethyl)oleamide | CHEMBL199649)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175109(N-(2,4-dimethoxyphenethyl)oleamide | CHEMBL199649)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Institute of Biomolecular Chemistry

Curated by ChEMBL
LigandPNGBDBM50175109(N-(2,4-dimethoxyphenethyl)oleamide | CHEMBL199649)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against rat brain FAAH by [14C]anandamide hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed