BDBM50184804 1-(2-fluorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazine::CHEMBL210717

SMILES Fc1ccccc1N1CCN(Cc2cnn(c2)-c2ccccc2)CC1

InChI Key InChIKey=UTUCAVNEOKJWJU-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50184804   

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184804(1-(2-fluorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)me...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184804(1-(2-fluorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)me...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2(short) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184804(1-(2-fluorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)me...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2(long) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184804(1-(2-fluorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)me...)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50184804(1-(2-fluorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)me...)
Affinity DataKi:  680nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in porcine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed