BDBM50185292 6-Benzyl-4-oxo-1,4-dihydroquinoline-3-carboxylic Acid EthylEster::6-benzyl-3-ethoxycarbonyl-4-quinolone::CHEMBL381059::ethyl 6-benzyl-4-oxo-1,4-dihydroquinoline-3-carboxylate
SMILES CCOC(=O)c1cnc2ccc(Cc3ccccc3)cc2c1O
InChI Key InChIKey=WQYYZNGOTUCWQX-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50185292
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair