BDBM50187439 1-(5-Methoxypyridin-3-yl)-[1,5]diazocane::1-(5-methoxypyridin-3-yl)-1,5-diazocane::CHEMBL378630
SMILES COc1cncc(c1)N1CCCNCCC1
InChI Key InChIKey=SHALYUZFJLUFSL-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50187439
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at human alpha4beta2 nAChR expressed in HEK293 cells assessed as intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair