BDBM50187442 1-(6-bromo-5-(vinyloxy)pyridin-3-yl)-1,5-diazocane::1-(6-bromo-5-vinyloxypyridin-3-yl)-[1,5]-diazocane::CHEMBL209618
SMILES Brc1ncc(cc1OC=C)N1CCCNCCC1
InChI Key InChIKey=BCTMPICFFTZGMY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50187442
Affinity DataIC50: 0.380nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.380nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Agonist activity at human alpha4beta2 nAChR expressed in HEK293 cells assessed as intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair