BDBM50190112 CHEMBL88808
SMILES NC(CCc1ccccc1)P(O)(=O)CC(Cc1ccc(O)cc1)C(O)=O
InChI Key InChIKey=STVSJGZHUJJREA-UHFFFAOYSA-N
Data 7 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50190112
TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of Plasmodium falciparum LAPMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of porcine APNMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of APN in porcine kidney using L-leucine p-nitroanilide as substrate preincubated for 60 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Inhibition of APA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Inhibition of porcine LAPMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
Wroclaw University Of Technology
Curated by ChEMBL
Wroclaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.04E+3nMAssay Description:Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
Wroclaw University Of Technology
Curated by ChEMBL
Wroclaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 6.47E+3nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair