BDBM50196452 (2S)-1-[(2S)-2-(1S)-3-oxocyclopentylcarboxamido]-3-(2-cyclohexyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide::CHEMBL376135
SMILES NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1cnc([nH]1)C1CCCCC1)NC(=O)[C@H]1CCC(=O)C1
InChI Key InChIKey=WDSXKLORUSKPMN-SNRMKQJTSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50196452
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]N(1)-Me-His-TRH from TRHR1More data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]N(1)-Me-His-TRH from TRHR2More data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair