BDBM50205833 CHEMBL222830::H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2
SMILES N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H]1CCCC[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)CNC1=O)C(N)=O
InChI Key InChIKey=RIGPFFUSPNYWOF-AFXVXQJMSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50205833
Affinity DataKi: 1.17nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.34nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 71.5nMAssay Description:Displacement of [3H]U69,593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.64nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 11.2nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair