BDBM50213650 CHEMBL233341::adamantan-1-yl-{2-(3,5-dimethyl-phenyl)-3-[(S)-1-methyl-2-(2-pyridin-4-yl-ethylamino)-ethyl]-1,4,6,7-tetrahydro-pyrrolo[3,2-c]pyridin-5-yl}-methanone
SMILES C[C@H](CNCCc1ccncc1)c1c2CN(CCc2[nH]c1-c1cc(C)cc(C)c1)C(=O)C12CC3CC(CC(C3)C1)C2
InChI Key InChIKey=DBZQPMXYZLHNKR-RPFINBQBSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50213650
Affinity DataKi: 1.5nMAssay Description:Displacement of [125I]-Tyr5, DLeu6, NMeLeu7, Pro-N-Et-GnRH from cloned rat GnRHRMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of GnRHR in rat pituitary cells assessed as inhibition of GnRH-stimulated LH releaseMore data for this Ligand-Target Pair
Affinity DataIC50: 546nMAssay Description:Inhibition of human GnRHR expressed in RBL cells assessed as inhibition of GnRH-stimulated [3H]-inositol phosphate hydrolysisMore data for this Ligand-Target Pair