BDBM50221623 2-(4-(methylsulfonyl)benzylsulfonyl)-6,7-dichloro-3-isopropylquinoxaline::CHEMBL251760

SMILES CC(C)c1nc2cc(Cl)c(Cl)cc2nc1S(=O)(=O)Cc1ccc(cc1)S(C)(=O)=O

InChI Key InChIKey=JQDWYVIABCGIHR-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50221623   

TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221623(2-(4-(methylsulfonyl)benzylsulfonyl)-6,7-dichloro-...)
Affinity DataIC50: 459nMAssay Description:Effect on augmentation of [125]GLP1 binding to human GLP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221623(2-(4-(methylsulfonyl)benzylsulfonyl)-6,7-dichloro-...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human GLP1 assessed as stimulation of cAMPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed