BDBM50222646 CHEMBL157917

SMILES COc1cc(CCCN(CCc2ccccc2)C(\S)=N\CCc2ccc(F)cc2)ccc1O

InChI Key InChIKey=SHLZVEQNSZIWEH-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50222646   

TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Seoul National University

Curated by ChEMBL

LigandBDBM50222646(CHEMBL157917)Copy SMILESCopy InChI

Affinity DataIC50: 5.10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/19/2018
Entry Details Article
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