BDBM50223013 CHEMBL400155::N-(cyclopropylmethyl)-3,6-dimethyl-5-(4-methylpyridin-2-yloxy)-N-propylpyrazin-2-amine

SMILES CCCN(CC1CC1)c1nc(C)c(Oc2cc(C)ccn2)nc1C

InChI Key InChIKey=WTNLDPKRAJDQIM-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50223013   

TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50223013(CHEMBL400155 | N-(cyclopropylmethyl)-3,6-dimethyl-...)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed