BDBM50228500 CHEMBL424597
SMILES Cn1c(nc2c(N)ncnc12)-c1ccccc1
InChI Key InChIKey=AWQBXXOPENTNRG-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50228500
Affinity DataKi: 23nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor transfected in CHO cell membranes after 3 hrs by microbeta scintillation counti...More data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor transfected in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 7.79E+3nMAssay Description:Antagonist activity at recombinant human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced adenylyl cyclase activi...More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A3 receptor transfected in CHO cell membranes after 3 hrs by microbeta scintillation counti...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))
Smith Kline & French Research
Curated by ChEMBL
Smith Kline & French Research
Curated by ChEMBL
Affinity DataKi: 2.41E+4nMAssay Description:Binding affinity (Ki) against human phosphatidylinositol 4-kinaseMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))
Smith Kline & French Research
Curated by ChEMBL
Smith Kline & French Research
Curated by ChEMBL
Affinity DataIC50: 3.49E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair