BDBM50232117 1-(5-tert-butyl-2-fluoro-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea::CHEMBL443586

SMILES CC(C)(C)c1ccc2c(c1)CC(F)C2NC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=GNRVWTIJRDMIID-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232117   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232117(1-(5-tert-butyl-2-fluoro-2,3-dihydro-1H-inden-1-yl...)Copy SMILESCopy InChI

Affinity DataIC50: 35nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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