BDBM50232118 (R)-1-(5-(1-hydroxy-2-methylpropan-2-yl)-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea::CHEMBL398856

SMILES CC(C)(CO)c1ccc2[C@@H](CCc2c1)NC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=YZZVNCQNKVSHRD-GOSISDBHSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232118   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232118((R)-1-(5-(1-hydroxy-2-methylpropan-2-yl)-2,3-dihyd...)Copy SMILESCopy InChI

Affinity DataIC50:  127nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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