BDBM50232140 CHEMBL255078::N-(5-bromo-2,3-dihydro-1H-inden-1-yl)-N'-1H-indazol-4-ylurea

SMILES O=C(Nc1cccc2[nH]ncc12)NC1CCc2cc(Br)ccc21

InChI Key InChIKey=NAEMZEHAVXOQSK-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232140   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232140(N-(5-bromo-2,3-dihydro-1H-inden-1-yl)-N'-1H-indazo...)Copy SMILESCopy InChI

Affinity DataIC50: 9nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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