BDBM50236536 CHEMBL4102553
SMILES Oc1ccc(cc1)-c1cnc2[nH]cc(-c3ccc(cc3)-c3nnn[nH]3)c2c1
InChI Key InChIKey=QZIYOWZOZNSBGJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50236536
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 172nMAssay Description:Inhibition of DYRK1B (unknown origin) using woodtide as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of DYRK1A (unknown origin) using woodtide as substrate after 10 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 416nMAssay Description:Inhibitory activity against Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataEC50: 8.50E+4nMAssay Description:Inhibition of CLK1 (unknown origin) using KKGRSRSRSRSRSR as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair